POSTER PRESANTATION
P-001 SYNTHESIS AND ANTITUMOR ACTIVITIES OF SOME 4,5-DIHIDRO-1-H1,2,4-TRIAZOL-5-ONES Aykut İkizler, Aysun İkizler, Haydar Yüksek, Mevlüt Serdar Departmant of Chemistry,Karadeniz Technical University, 61080, Trabzon, Turkey. P-002 SYNTHESIS AND ANTİCANCER ACTIVITIES OF SOME 3,4-DISUBSTITUTED-4,5-DIHYDRO-1H-1,2,4-TRIAZOL-5-ONES Aykut İkizler, Haydar Yüksek, Şule Bahçeci Departmant of Chemistry,Karadeniz Technical University, 61080, Trabzon, Turkey. P-003 DETERMINATION OF PHENYTOIN SODIUM IN SOLID DOSAGE FORMS VIA HPLC METHOD Seyhan Ersan, Ahmet Üngörmüş, Tuncel Özden Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Gazi, 06330 Hipodrom Ankara Turkey P-004 SYNTHESIS OF HYDRAZONES OF [(3-SUBSTITUED-1,2,4-TRIAZOLYL-5-THIO)ACETYL] HYDRAZINE Seyhan Ersan and Sultan Nacak Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Gazi, 06330 Hipodrom Ankara Turkey P-005 QANTITATIVE HIGH PERFORMANCE LIQUID CHROMATOGRAPHIC ANALYSIS OF FAMOTIDINE IN PHARMACEUTICAL DOSAGE FORMS B.Cakır, A.U. Tosun, M.F. Sahin P-006 ANALYTICAL RESOLUTION OF 4-ARYL-1,2,3,4,5,6,7,8-OCTA-HYDROQUINAZOLINE-2-THIONES USING A CELLULOSE CHIRAL STATIONARY PHASE Selma Saraç, Mine Yarım, Mevlüt Ertan Hacettepe University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, 06100 Ankara-Turkey P-007 SOME AZOLYLTHIOACETAMİDES AND THEIR ANALGESİC AND ANTIINFLAMMATORY ACTİVİTİES Rahime Şimşek*, Pelin Kelicen**, Hülya Akgün*, Cihat Şafak*, Rümeysa Demirdamar** * Dept. of Pharm.Chemistry, Fac. of Pharmacy, Hacettepe University,Ankara-TURKEY ** Dept. of Pharmacology, Fac. of Pharmacy, Hacettepe University, Ankara-TURKEY P-008 NEW 2,6,6-TRIMETHYL-3-ACYL-4-ARYL-5-OXO-1,4,5,6,7,8-HEXAHYDRQUINOLINE DERIVATIVES Yeşim Altaş, Rahime Şimşek, Cihat Şafak Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Hacettepe University, Ankara-TURKEY P-009 TITRIMETRIC DETERMINATION OF ACTIVE COMPOUNDS IN CANNABIS SATIVA WITH SeO3-2 Hasan Aydın Gazi Un. Fen-Edebiyat Fakültesi Kimya Bölümü P-010 ONE FLAVONOID FROM VERBASCUM ANCYRITANUM BORNM. Yılmaz Yıldırır* and Naki Colak Gazi University, Science and Arts Faculty, Department of Chemistry, Teknikokullar, Ankara,06500, Turkey P-011 SYNTHESIS AND ANTICANCER AND ANTI-HIV ACTIVITIES OF SOME PYRAZINO-BENZIMIDAZOLE DERIVATIVES Şeref Demirayak, Usama A.Mohsen University of Anadolu, Faculty of Pharmacy, Dept. of Pharmaceutical Chemistry, Eskişehir, Türkiye P-012 SYNTHESIS AND ANTIBACTERIAL EVOLUTION OF SOME ETHYL 1-ARYLOXYACETYLAMINO-5-ARYLPYRROLE-3-CARBOXYLIC ACID DERIVATIVES Şeref Demirayak1, Ahmet Ç. Karaburun1, Nuri Kiraz2 1Unıversity of Anadolu, Faculty of Pharmacy, Dept. of Pharmaceutical Chemistry, Eskişehir, Türkiye 2Unıversity of Osmangazi, Faculty of Medicine, Dept. of Microbiology, Eşkişehir, Türkiye. P-013 SYNTHESIS AND VASODILATORY ACTIVITY OF SOME 1-BENZIMIDAZOLYLMETHYL-TRIAZOLE DERIVATIVES Şeref Demirayak1, Kadriye Benkli1, Usama A. Mohsen1,Özlem Batu2, Kevser Erol2 1University of Anadolu, Faculty of Pharmacy, Dept. of Pharmaceutical Chemistry, Eskişehir, Türkiye 2University of Osmangazi, Faculty of Medicine, Dept. of Pharmacology, Eskişehir, Türkiye P-014 QUANTITATIVE DETERMINATION OF FLUCONAZOLE BY INFRARED SPECTROPHOTOMETRY Okan Atay*, Fatmagül Selçuk** *Gazi Üniversitesi Eczacılık Fakültesi Farmasötik Kimya A.B.D. Ankara **Abdi İbrahim İlaç Sanayii A.Ş. Vefa- İstanbul P-015 SYNTHESIS AND STRUCTURAL ELUCIDATION OF SOME 3-(2-and/or 4-PYRIDYLETHYL)BENZOXAZOLINONES Nesrin Gökhan, Hakkı Erdoğan Hacettepe University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry 06100 Ankara Turkey P-016 STUDIES ON THE SYNTHESIS OF SOME TRIAZOLES AND TRIAZOLO-TIADIAZINES G.Turan-Zitouni, Z.A. Kaplancıklı Anadolu University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry 26470-Eskişehir Turkey P-017 MODULATION OF OOIOID RECEPTOR BINDING BY ARACHIDONIC ACID AND LYSOPHOSATIDIC ACID Serpil Apaydın, Hüseyin Avni Öktem Depertment of Biology, Middle East Tecnical University, 06531 Ankara, Turkey P-018 SYNTHESİS AND HYPNOTIC ACTIVITY OF NEW 2-THIOXO-4,5-İMİDAZOLİDİNEDİONE AND 4-THIAZOLIDINONE DERIVATIVES N.Ergenç1, G.Çapan1, N.S.Günay1, S. Özkırımlı1, M. Güngör2 1 University of İstanbul, Faculty of Pharmacy, Department of pharmaceutical Chemistry,34452 İstanbul,2 İstanbul Faculty of Medicine, Department of Pharmacology 34390 İstanbul-TURKEY P-019 SYNTHESIS AND ANTIMICROBIAL ACTIVITIES OF SOME 2-[(4-CARBETHOXY-METHYLTHIAZOL-2-YL)IMINO]-4-THIAZOLIDINONE DERIVATIVES Ö.Ateş*, H.Altıntaş*, G.Ötük**, A.S.Birteksöz**, *University of Istanbul, Faculty of Pharmacy, Dept. of Pharmaceutical Chemistry **Dept.of Pharmaceutical Microbiology P-020 SYNTHESIS AND ANTIMICROBIAL ACTIVITIES OF SOME 5-ARYL-2-[(N,N-DISUBSTITUTEDTHIOCARBAMOYLTHIO)ACYLAMINO]-1,3,4-OXADIAZOLES. Ö. Ateş*, A. Kocabalkanlı*, N. Cesur*, G. Ötük** *University of Istanbul, Faculty of Pharmacy, Dept. of Pharmaceutical Chemistry **Dept. of Pharmaceutical Microbiolgy. P-021 SYNTHESIS AND ANTIMICROBIAL ACTIVITIES OF SOME N,N-DISUBSTITUTED- CARBAMODITHIOIC ACID ESTERS S. Özkırımlı*, T.İ. Apak*, G. Ötük**, A.S. Birteksöz** * University of Istanbul, Faculty of Pharmacy, Dept.of Pharmaceutical Chemistry **Dept. of Pharmaceutical Microbiology. P-022 SOME IMIDAZO[1,2-a]PYRIDINE DERIVATIVES AS POSSIBLE ANTIMYCOBACTERIALS Z. Cesur, N. Cesur University of Istanbul, Faculty of Pharmacy, Dept. of Pharmaceutical Chemistry P-023 THE ADDITION PRODUCTS OF THIOSALICYCLIC ACID AND b-NITROSTYRENES AND THEIR ANTIMICROBIAL ACTIVITIES Mehtap Gökçe1, Berrin Özçelik2, Erdoğan Berçin1 1Gazi University Faculty of Pharmacy Department of Pharmaceutical Chemistry 2Gazi University Faculty of Pharmacy Department of Microbiology 06330-Hipodrum-Ankara P-024 SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF 6-FLAVONE CARBOXALDEHYDE OXIME ETHER DERIVATIVES G. Ayhan Kılcıgil1, O. Bozdağ1, M. Tunçbilek1, N. altanlar2, R. Ertan1 Ankara University, 1Deparment of Pharmaceutical Chemistry, 2Deparment of Microbiology, Faculty of Pharmacy, 06100-Tandoğan,Ankara, Turkey P-025 NEW FLAVONYL OXIME-ETHER DERIVATIVES: SYNTHESIS AND ANTIMICROBIAL ACTIVITY M.Tunçbilek1 , O. Bozdağ1, G. A. Kılcıgil1, N. Altanlar2, R. Ertan1. Ankara University, Depertmant of Pharmaceutıcal Chemistry, Depertmant of Mıcrobıology, Faculty of Pharmacy, 06100-Tandoğan, Ankara, Turkey P-026 STUDIES ON THE SYNTHESIS AND BIOLOGICAL ACTIVITY OF SOME NEW OXIME-ETHER DERIVATIVES O.Bozdağ1, G. A. Kılcıgil1, M. Tunçbilek1, N. Altanlar2, R. Ertan1. Ankara University, Depertmant of Pharmaceutıcal Chemistry, Depertmant of Mıcrobıology, Faculty of Pharmacy, 06100-Tandoğan, Ankara, Turkey P-027 QSAR ANALYSIS OF SOME NOVEL SUBSTITUTED BENZOXAZOLES AGAINST C.ALBICANS USING THE PLS REGRESSION METHOD Özlem Temiz*, İlkay Ören*, Yılmaz Akdi** and Levent Özbek** *Ankara University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Tandoğan, 06100 Ankara (Turkey) ** Ankara University, Faculty of Science, Department of Statistic, Tandoğan, 06100 Ankara (Turkey) P-028 SYNTHESIS AND IN VITRO MICROSOMAL METABOLISM OF 4-ETHYL-5-(4-FLUOROPHENYL)-2,4-DIHYDRO-3H-THIONE AND ITS POTENTIAL METABOLITES N. Gülerman, S. Rollas and M. Ülgen Marmara University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry 08010 Haydarpaşa, Istanbul,Turkey. P-029 REDUCTIVE CLEAVAGE OF SOME COMPOUNDS CONTAINING TRIAZENE FUNCTIONAL GROUP WITH HYDRAZINE HYDRATE S.Rollas, S.Ünsalan, E.E. Oruç and S. Büyüktimkin Marmara University, Faculty of Pharmacy 81010, Haydarpaşa, İstanbul,TURKEY KansasUniversity, Pharmaceutical Chemisty12065 Constant Avenue Lawrence, KS 660 45, USA P-030 SYNTHESIS AND STRUCTURE ELUCIDATION OF SOME NEW HYDRAZONE AND 3-ACETYL-2,5-DISUBSTITUTED-1,3,4-OXADIAZOLINES H.Neşe Doğan, Arzu Duran, Sevim Rollas Marmara University, Faculty of Pharmacy 81010, Haydarpaşa, İstanbul,TURKEY P-031 THIAZOLO[3,2-b]-1,2,4-TRIAZOLE(6H)-ONES: SYNTHESIS AND EVALUATION OF ANTIINFLAMMATORY ACTIVITY B. Tozkoparan1, G. Ayhan Kılcıgil2, R. Ertan2, M. Ertan1, S. Özbey, E. Kendi3, P. Kelicen, R. Demirdamar4 1Hacettepe Univ., Faculty of Pharmacy, Dept. of Pharm. Chemistry 06100 2Ankara Univ., Faculty of Pharmacy, Dept. of Pharm. Chem. 06100 3Hacettepe Univ., Dept. of Physics Engineering 06532 4Hacettepe Univ., Faculty of Pharmacy, Dept. of Pharmacology 06100 Ankara-Turkey P-032 SYNTHESIS OF SOME NEW PYRAZOLINE DERIVATIVES WITH BIOLOGICAL ACTIVITIES G. Öztürk, M. Aytemir, E. Palaska, D. Erol Hacettepe Univ., Faculty of Pharmacy, Pharmaceutical Chemistry Dept. 06100 Ankara-Turkey P-033 SYNTHESIS AND ANALGESIC & ANTIINFLAMMATORY ACTIVITIES OF SOME NEW SUBSTITUTED 4-PYRIDONE DERIVATIVES Gülcan Öztürk*, T. Uzbay**, D. Erol* *Hacettepe Univ. Faculty of Pharmacy, Pharmaceutical Chemistry Dept. 06100 Ankara-Turkey **Military Medical Academy of Gulhane, Department Pharmacology, Etlik, Ankara P-034 SYNTHESIS,CHARACTERIZATION AND ANTIMICROBIAL EVALUATION OF 4-ARYLHYDRAZONO-2-PYRAZOLINE-5-ONES Ş.G.Küçükgüzel1,S.Rollas1,H.Erdeniz2 and M.Kiraz2 1Marmara Universith, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Tıbbiye cad.81010,Haydarpaşa, İstanbul, Türkiye 2University of İstanbul, Faculty of Medicine, Center for Research and Application of Culture Collections of Microorganisms, Çapa, İstanbul, Türkiye P-035 EFFECT OF NITROGEN pKa ON THE MICROSOMAL OXIDATION OF N-BENZYLIC HETEROCYCLES İ. Küçükgüzel1, M. Ülgen, J. W. Gorrod2 1 Marmara University, Faculty of Pharmacy, Department of Pharmaceutical Chemistry, Tıbbıye cad. 81010 Haydarpaşa, İstanbul, Türkiye. 2 Chelsea Department of Pharmacy, King’s College London, University of London, Manresa Road, London, SW3 6LX, UK. P-036 NEW 4-PYRIDONE DERIVATIVES AS ANALGESIC AGENTS M. D., Aytemir*,T., Uzbay**, D.D., Erol* *Hacettepe Univ., Faculty of Pharmacy, Pharmaceutical Chemistry Dept., 06100 Ankara-Turkey **Military medical academy of Gülhane, Department Pharmacology, Etlik, Ankara P-037 STUDIES ON PYRAZOLINE DERIVATIVES Ozan Ruhoğlu, A. Altan Bilgin Hacettepe Univ., Faculty of Pharmacy, Pharmaceutical Chemistry Dept., 06100 Ankara-Turkey P-038 SYNTHESIS AND ANTICONVULSANT ACTIVITY OF SOME NEW NAFİMİDON OXİME AND OXİME ETHERS DERIVATIVES Arzu Karakurt, Sevim Dalkara Hacettepe Univ., Faculty of Pharmacy, Pharmaceutical Chemistry Dept., 06100 Ankara-Turkey P-039 ALKALOID WOODININE Siavoush Mahboobi Department of Pharmaceutical Chemistry, University, D-93040 Regensburg, Germany P-040 AZO-, NEUTROCYANINE- AND AZAMETHINE-DYES WITH 3-AMINOHODANINE AS CORE STRUCTURE. W. Hanefeld, H. Euler and M. Schlitzer Inst. f. Pharmazeut. Chemie, Philipps-Universität, Marbacher Weg 6, D-35032 Marburg, Germany P-041 CAPILLARY ELECTROPHORESIS SEPARATION OF ASPARTYL- AND GLUTAMYL-DIPEPTIDES Gerhard K. E. Scriba Departman of Pharmaceutical Chemistry, University of Münster, Hittorfstrasse 58-62, 41849 Münster, Germany. P-042 SYNTHESIS OF SOME 3-ETHANONE-2-BENZOXAZOLINON DERIVATIVES AND THEIR ANTIMICROBIAL ACTIVITIES Ünsal Çalış*, Dilek Demir Erol*, Nuran Yuluğ** *Hacettepe University, Faculty of Pharmacy, Pharmaceutical Chemistry Department, Ankara (Turkey) **9 Eylül University, Medical Faculty, Microbiology Depertment, İzmir (Turkey)